AM580
Product Name : AM580Description:AM-580 is a potent RARalpha agonist. AM580 has powerful and selective cyto-differentiating effects on acute promyelocytic leukemia cells. AM580 inhibited the wnt pathway, measured by loss of…
M2e, human TFA
Product Name : M2e, human TFADescription:M2e, human TFA, consisting of the 23 extracellular residues of M2 (the third integral membrane protein of influenza A), has been remarkably conserved in all…
Zinterol
Product Name : ZinterolDescription:Zinterol (MJ 9184) is a potent and selective β2-adrenoceptor agonist. Zinterol increases ICa in a concentration-dependent manner with an EC50 of 2.2 nM.CAS: 37000-20-7Molecular Weight:378.49Formula: C19H26N2O4SChemical Name:…
CYT387 (sulfate salt)
Product Name : CYT387 (sulfate salt)Description:Momelotinib (CYT387, LM-1149 , CYT11387) is an ATP-competitive inhibitor of JAK1/JAK2 with IC50 of 11 nM/18 nM, ~10-fold selectivity versus JAK3. Momelotinib (CYT387) induces apoptosis…
AP-1/NF-κB activation inhibitor 1
Product Name : AP-1/NF-κB activation inhibitor 1Description:AP-1/NF-κB activation inhibitor 1 is a potent AP-1 and NF-κB mediated transcriptional activation inhibitor (IC50=1 μM), without blocking basal transcription driven by the β-actin…
Retrobradykinin
Product Name : RetrobradykininDescription:Retrobradykinin has the reverse sequence of Bradykinin (HY-P0206). Retrobradykinin exhibits no kinin activity and can be used as a negative control for Bradykinin.CAS: 5991-13-9Molecular Weight:1060.21Formula: C50H73N15O11Chemical Name:…
Ethyl nonanoate
Product Name : Ethyl nonanoateDescription:Ethyl nonanoate is a rich ester in spirits and its presence is commonly related to the pleasant fruity bouquet of alcoholic beverages. Ethyl nonanoate is an…
Midostaurin-D5
Product Name : Midostaurin-D5Description:Midostaurin-D5 (PKC412-D5) is a deuterium labeled Midostaurin. Midostaurin is a multi-targeted protein kinase inhibitor which inhibits PKCα/β/γ, Syk, Flk-1, Akt, PKA, c-Kit, c-Fgr, c-Src, FLT3, PDFRβ and…
BAY 1436032
Product Name : BAY 1436032Description:BAY-1436032 is a highly selective, potent and orally available inhibitor of mutant Isocitrate Dehydrogenase 1 (mIDH1). It is a double-digit nanomolar and selective pan-inhibitor of the…
EMD638683 (S)
Product Name : EMD638683 (S)Description:EMD638683 S-Form is the S-form of EMD638683. EMD638683 is a highly selective SGK1 inhibitor with IC50 of 3 μM.CAS: 1184940-46-2Molecular Weight:364.34Formula: C18H18F2N2O4Chemical Name: (2S)-2-(3,5-difluorophenyl)-N'-(2-ethyl-4-hydroxy-3-methylbenzoyl)-2-hydroxyacetohydrazideSmiles : CC1C(O)=CC=C(C=1CC)C(=O)NNC(=O)(O)C1C=C(F)C=C(F)C=1InChiKey:…